Briquilimab Antibody Delivers Rapid, Lasting Relief in Chronic Urticaria Trials (targeting KIT (CD117)

Jasper Therapeutics announced promising updated clinical data on January 8, 2026, for briquilimab, a monoclonal antibody targeting KIT (CD117) to deplete mast cells and treat mast cell-driven conditions like chronic spontaneous urticaria (CSU) and chronic inducible urticaria (CIndU).

Key highlights include rapid and durable symptom relief, measured by the Urticaria Activity Score over 7 days (UAS7, where 0 indicates complete response):

In additional BEACON participants (240mg loading dose followed by 180mg every 8 week) 83% achieved complete response (UAS7=0) by week 3, and 67% maintained it at week 12.

The dosing is every 2 months.

For CIndU patients, 65% showed complete or partial response at 16 weeks (after the second dose).

The therapy demonstrated a favorable safety profile, with no dose-limiting toxicities.

The data reaffirm briquilimab's potential for rapid, durable control in CSU. This is a new mast cell-targeted approach in addressing unmet needs in chronic urticaria.

Over 20 companies are advancing chronic urticaria trials, with mentions of: 

- oral KIT inhibitors

- barzolvolimab (KIT inhibitor) progressing in Phase 3 for CSU and inducible forms like cold urticaria/symptomatic dermographism 

- oral MRGPRX2 inhibitors focused on CSU (and potential in asthma, prurigo nodularis)


Chronic Urticaria Treatment Options (click to enlarge the image). 

References:

https://ir.jaspertx.com/news-releases/news-release-details/jasper-therapeutics-reports-positive-updated-data-briquilimab